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GPCR Weekly News

January 23, 2025

GPCR Weekly: Key Activating Interactions, Lysosomal Signaling & a Dash of Pheromones! ➼ Jan 13 - 19, 2025

January 17, 2025

The GPCR Momentum: Keeping the Discoveries Rolling! → Jan 6 - 12, 2025

January 9, 2025

Back to GPCR Business: Starting the Year with a Bang! ✴︎ Dec 16, 2024 - Jan 5, 2025

Contributors Articles

John Teye Azietaku

Reflections on My PhD Journey: Lessons Learned

Cam Sinh Lu

Harnessing Deep Mutational Scanning for Enhanced Drug Discovery

John Teye Azietaku

Class B1 GPCR Dimerization: Unveiling Its Role in Receptor Function and Signaling

GPCR Industry News

January 23, 2025

Computational tool designs proteins with water-mediated interactions in mind

January 21, 2025

AI, data, and the acceleration of drug discovery

January 24, 2025

Research could lead to better medicines and new tools in synthetic biology

Call for GPCR Papers

November 1, 2024

Emerging Voices in GPCR Biology in Special Issue of Molecular Pharmacology

September 27, 2023

opnMe GPCR Route 66+ project

March 31, 2023

GPCRs: Signal Transduction

Adhesion GPCRs

January 9, 2025

N-terminal fragment shedding contributes to signaling of the full-length adhesion receptor ADGRL3

January 1, 2025

Novel Isoforms of Adhesion G Protein-Coupled Receptor B1 (ADGRB1/BAI1) Generated from an Alternative Promoter in Intron 17

GPCR Activation and Signaling

January 21, 2025

GRK5 is required for adipocyte differentiation through ERK activation

January 20, 2025

GPCR oligomerization across classes: A2AR-mediated regulation of mGlu5R activation

January 13, 2025

Key Interaction Changes Determine the Activation Process of Human Parathyroid Hormone Type 1 Receptor

GPCR Binders, Drugs, and more

January 24, 2025

Novel tertiary diarylethylamines as functionally selective agonists of the kappa opioid receptor

January 10, 2025

A lipidated peptide derived from the C-terminal tail of the vasopressin 2 receptor shows promise as a new β-arrestin inhibitor

December 18, 2024

Integrated NMR-crystallography-computational approach for molecular recognition studies of human Gαi3 protein by a small molecule inhibitor

GPCRs in Cardiology, Endocrinology, and Taste

January 7, 2025

LGR4 is essential for maintaining β-cell homeostasis through suppression of RANK

November 28, 2024

Metabolic control of Luteinizing Hormone-responsive ovarian steroidogenesis

November 25, 2024

Cardiovascular Complications and Their Association With Short- and Long-Term Outcomes in Patients With Multiple Myeloma and Lymphoma Undergoing Chimeric Antigen Receptor T-Cell Therapy

FRPR-1, a G protein-coupled receptor (GPCR) in the FMRFamide-related peptide receptor family, modulates larval development as a receptor candidate of the FMRFamide-like peptide FLP-1 in Caenorhabditis elegans

January 1, 2025

Comparing adenosine A2A receptor modulation of cannabinoid CB1 receptor-mediated inhibition of GABA and glutamate release in rodent striatal nerve terminals

December 18, 2024

CaV3.2 T-type calcium channels contribute to CGRP- induced allodynia in a rodent model of experimental migraine

GPCRs in Oncology and Immunology

January 13, 2025

G protein-coupled purinergic P2Y receptors in infectious diseases

January 6, 2025

A New Strategy in Modulating the Protease-Activated Receptor 2 (Par2) in Autoimmune Diseases

December 19, 2024

The development of murine bone marrow-derived mast cells expressing functional human MRGPRX2 for ex vivo and in vivo studies

Methods & Updates in GPCR Research

January 17, 2025

Development of a yeast-based sensor platform for evaluation of ligands recognized by the human Free Fatty Acid 2 Receptor

January 8, 2025

The influence of phosphoinositide lipids in the molecular biology of membrane proteins: recent insights from simulations

December 16, 2024

Development of a Class A/B Hybrid GPCR System for the Proximity-Assisted Screening of GPCR Ligands

Reviews, GPCRs, and more

January 24, 2025

An update on regulation and function of G protein-coupled receptors in cancer: A promising strategy for cancer therapy

January 24, 2025

Early intervention with daratumumab improves survival for patients with high-risk smouldering myeloma

January 20, 2025

GPCR Biosensors to Study Conformational Dynamics and Signaling in Drug Discovery

Structural and molecular insights into GPCR function

January 17, 2025

Molecular architecture of human LYCHOS involved in lysosomal cholesterol signaling

January 18, 2025

Unraveling the Molecular Architecture of Mosquito D1-Like Dopamine Receptors: Insights Into Ligand Binding and Structural Dynamics for Insecticide Development

January 17, 2025

Cryo-EM reveals cholesterol binding in the lysosomal GPCR-like protein LYCHOS

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