GPCR News 

Identification and functional characterization of the sulfakinin and sulfakinin receptor in the...

Sweet taste receptor agonists attenuate macrophage IL‐1β expression and eosinophilic inflammation...

Dynamic recognition of naloxone, morphine and endomorphin1 in the same pocket of µ-opioid receptors

Functional Characterization of the Venus Flytrap Domain of the Human TAS1R2 Sweet Taste Receptor

Combined docking and machine learning identify key molecular determinants of ligand pharmacological

Divergent roles for the gut intraepithelial lymphocyte GLP-1R in control of metabolism, microbiota..

Targeting mGluR2/3 for treatment of neurodegenerative and neuropsychiatric diseases

Identification of hub genes in the subacute spinal cord injury in rats

Endogenous ligand recognition and structural transition of a human PTH receptor

CD28 and chemokine receptors: Signalling amplifiers at the immunological synapse

Serotonin Receptor 5-HT2A Regulates TrkB Receptor Function in Heteroreceptor Complexes

PAR-Induced Harnessing of EZH2 to β-Catenin: Implications for Colorectal Cancer

Endocannabinoid System in the Neuroendocrine Response to Lipopolysaccharide-induced Immune Challenge

Isoform-and ligand-specific modulation of adhesion GPCR ADGRL3/Latrophilin3 by a synthetic binder

Arginine 125 Is an Essential Residue for the Function of MRAP2

Immunomodulatory Role of Neuropeptides in the Cornea

GPR108 is required for gambogic acid inhibiting NF-κB signaling in cancer

Dynamics of tumor-associated macrophages in a quantitative systems pharmacology model of...

GPCR kinase phosphorylation of distal C-tail sites specifies βarrestin1-mediated signaling by...

The Impact of CB1 Receptor on Nuclear Receptors in Skeletal Muscle Cells