GPCR News 

Endosomal parathyroid hormone receptor signaling

Targeting CXCR1 and CXCR2 receptors in cardiovascular diseases

Allosteric modulation of GPCRs: From structural insights to in silico drug discovery

Structural perspectives on the mechanism of signal activation, ligand selectivity and allosteric...

Identification of A2BAR as a potential target in colorectal cancer using novel fluorescent GPCR...

GPCR Agonist-to-Antagonist Conversion: Enabling the Design of Nucleoside Functional Switches for...

Endogenous ligand recognition and structural transition of a human PTH receptor

Coincident Regulation of PLCβ Signaling by Gq-Coupled and μOpioid Receptors Opposes Opioid- Mediated

Intermolecular Interactions in G Protein-Coupled Receptor Allosteric Sites at the Membrane Interface

ADGRL3 genomic variation implicated in neurogenesis and ADHD links functional effects to the...

Adenosine receptor signalling in Alzheimer's disease

Glucagon receptor-mediated regulation of gluconeogenic gene transcription is endocytosis-dependent..

Keratinocyte-derived defensins activate neutrophil-specific receptors Mrgpra2a/b to prevent skin...

Mechanistic Understanding of the Palmitoylation of Go Protein in the Allosteric Regulation of...

Production of human A2AAR in lipid nanodiscs for 19F-NMR and single-molecule fluorescence...

Activation of GPR183 by 7 α,25-Dihydroxycholesterol Induces Behavioral Hypersensitivity through...

Use of CRISPR/Cas9-edited HEK293 cells reveals that both conventional and novel protein kinase C...

N-Acyl Amides from Neisseria meningitidis and Their Role in Sphingosine Receptor Signaling

Function and structure of bradykinin receptor 2 for drug discovery

Specific Functions of Melanocortin 3 Receptor (MC3R)