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Dr. GPCR News
Aug 24, 20221 min read
Learn about Dr. GPCR Ecosystem!
💻Did you know that Dr. GPCR is much more than a podcast? Come check out the brand new Dr. GPCR Ecosystem and explore its benefits! We...
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Dr. GPCR News
Aug 23, 20221 min read
Dr. GPCR Summit is FREE for Ecosystem site members!
📢 Did you know that this 3rd Edition of the Dr. GPCR Summit is totally FREE for our Ecosystem site members? Join us and become a site...
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GPCR News
Aug 1, 20221 min read
Opioid Ligands Addressing Unconventional Binding Sites and More Than One Opioid Receptor Subtype
August 2022 "Opioid receptors (ORs) represent one of the most significant groups of G-protein coupled receptor (GPCR) drug targets and...
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GPCR News
Aug 1, 20221 min read
In vitro assays for the functional characterization of (psychedelic) substances at the serotonin...
August 2022 In vitro assays for the functional characterization of (psychedelic) substances at the serotonin receptor 5-HT2A R...
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GPCR News
Jul 31, 20221 min read
Activation of the human chemokine receptor CX3CR1 regulated by cholesterol
August 2022 "As the only member of the CX3C chemokine receptor subfamily, CX3CR1 binds to its sole endogenous ligand CX3CL1, which shows...
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GPCR News
Jul 31, 20221 min read
Murine bone marrow macrophages and human monocytes do not express atypical chemokine receptor 1
August 2022 "The atypical chemokine receptor 1 (ACKR1) was discovered on erythrocytes as the Duffy blood group antigen ( Cutbush et al.,...
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GPCR News
Jul 31, 20221 min read
Dopamine D 1 receptor-mediated β-arrestin signaling: Insight from pharmacology, biology, behavior...
August 2022 Dopamine D 1 receptor-mediated β-arrestin signaling: Insight from pharmacology, biology, behavior, and neurophysiology "The...
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GPCR News
Jul 31, 20221 min read
Production of human A2AAR in lipid nanodiscs for 19F-NMR and single-molecule fluorescence...
August 2022 Production of human A 2A AR in lipid nanodiscs for 19 F-NMR and single-molecule fluorescence spectroscopy "We describe...
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GPCR News
Jul 31, 20221 min read
A correlation study of adhesion G protein-coupled receptors as potential therapeutic targets in...
August 2022 A correlation study of adhesion G protein-coupled receptors as potential therapeutic targets in Uterine Corpus Endometrial...
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GPCR News
Jul 31, 20221 min read
8th RSC / SCI symposium on GPCRs in Medicinal Chemistry. October 5-7, 2022, Verona, Italy
August 2022 "GPCRs in Medicinal Chemistry Event 8th RSC / SCI symposium on GPCRs in Medicinal Chemistry Dates Wednesday-Friday, 5th-7th...
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GPCR News
Jul 31, 20221 min read
Structure Therapeutics Extends Financing, Advances Diabetes and Obesity Clinical Program and...
August 2022 Structure Therapeutics Extends Financing, Advances Diabetes and Obesity Clinical Program and Changes Name from ShouTi "San...
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GPCR News
Jul 31, 20221 min read
Therapeutic validation of an orphan G protein-coupled receptor: The case of GPR84
August 2022 "Despite the importance of members of the GPCR superfamily as targets of a broad range of effective medicines many GPCRs...
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GPCR News
Jul 31, 20221 min read
Jan Steyaert Named 2022 Jacob and Louise Gabbay Award Winner
August 2022 "August 12, 2022.- Jan Steyaert, scientific director of the VIB-VUB Center for Structural Biology, Vlaams Instituut...
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GPCR News
Jul 31, 20221 min read
Structural basis of GPCR coupling to distinct signal transducers: implications for biased signaling
August 2022 "Three classes of G-protein-coupled receptor (GPCR) partners - G proteins, GPCR kinases, and arrestins - preferentially bind...
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GPCR News
Jul 31, 20221 min read
Amgen to Acquire Chemocentryx for $4 Billion in Cash
August 2022 "THOUSAND OAKS, Calif. and SAN CARLOS, Calif., Aug. 4, 2022 /PRNewswire/ -- Amgen (NASDAQ: AMGN) and ChemoCentryx, Inc.,...
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GPCR News
Jul 31, 20221 min read
Deciphering the signaling mechanisms of β-arrestin1 and β-arrestin2 in regulation of cancer cell...
August 2022 Deciphering the signaling mechanisms of β-arrestin1 and β-arrestin2 in regulation of cancer cell cycle and metastasis...
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GPCR News
Jul 31, 20221 min read
GPCRs steer G i and G s selectivity via TM5-TM6 switches as revealed by structures of serotonin...
August 2022 GPCRs steer G i and G s selectivity via TM5-TM6 switches as revealed by structures of serotonin receptors "Serotonin (or...
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GPCR News
Jul 31, 20221 min read
Addex and Indivior Extend GABAB Positive Allosteric Modulator Research Collaboration for...
August 2022 Addex and Indivior Extend GABAB Positive Allosteric Modulator Research Collaboration for Substance Use Disorders "Geneva,...
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GPCR News
Jul 31, 20221 min read
Gαs and Gαq/11 protein coupling bias of two AVPR2 mutants (R68W and V162A) that cause nephrogenic di
August 2022 Gαs and Gαq/11 protein coupling bias of two AVPR2 mutants (R68W and V162A) that cause nephrogenic diabetes insipidus...
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