GPCR News 

The Adhesion GPCR VLGR1/ADGRV1 Regulates the Ca2+ Homeostasis at Mitochondria-Associated ER Membrane

Mechanism of enhanced sensitivity of mutated β-adrenergic-like octopamine receptor to amitraz in...

Focusing on the role of secretin/adhesion (Class B) G protein-coupled receptors in placental...

Enhanced membrane binding of oncogenic G protein αqQ209L confers resistance to inhibitor YM-254890

N-terminal alterations turn the gut hormone GLP-2 into an antagonist with gradual loss of GLP-2 ...

GPR15 expressed in T lymphocytes from RA patients is involved in leukocyte chemotaxis to the...

PH-Binding Motif in PAR4 Oncogene: From Molecular Mechanism to Drug Design

Single-molecule counting applied to the study of GPCR oligomerization

Membrane Lipids Are an Integral Part of Transmembrane Allosteric Sites in GPCRs: A Case Study of...

Dopamine activates astrocytes in prefrontal cortex via α1-adrenergic receptors

Novel Therapies for Cardiometabolic Disease: Recent Findings in Studies with Hormone...

Advancements in G protein-coupled receptor biosensors to study GPCR-G protein coupling

Network pharmacological investigation into the mechanism of Kaixinsan powder for the treatment of...

Diversification of PAR signaling through receptor crosstalk

Comparative study of neuropeptide signaling systems in Hemiptera

Lysosomal GPCR-like protein LYCHOS signals cholesterol sufficiency to mTORC1

Regulation of pulmonary surfactant by the adhesion GPCR GPR116/ADGRF5 requires a tethered agonist...

A cryptic mode of GPCR regulation revealed

Design and validation of recombinant protein standards for quantitative Western blot analysis of...

Genome-scale CRISPR screening reveals that C3aR signaling is critical for rapid capture of fungi...

Successful prednisolone or calcimimetic treatment of acquired hypocalciuric hypercalcemia caused...

Developing the Cannabinoid Receptor 2 (CB2) pharmacopoeia: past, present, and future

The microglial endocannabinoid system similarly regulated by lipopolysaccharide and interferon gamma

Co-activation of GPCRs facilitate GIRK-dependent current