Blog: Blog2

GPCR News

Sep 30, 20221 min read

Identification of A2BAR as a potential target in colorectal cancer using novel fluorescent GPCR...

October 2022 Identification of A2BAR as a potential target in colorectal cancer using novel fluorescent GPCR ligands "G-protein coupled...

Aug 31, 20221 min read

A2B Adenosine Receptor Enhances Chemoresistance of Glioblastoma Stem-Like Cells under Hypoxia: New..

September 2022 A2B Adenosine Receptor Enhances Chemoresistance of Glioblastoma Stem-Like Cells under Hypoxia: New Insights into MRP3...

Aug 31, 20221 min read

Combined docking and machine learning identify key molecular determinants of ligand pharmacological

September 2022 "G protein‐coupled receptors (GPCRs) are valuable therapeutic targets for many diseases. A central question of GPCR drug...

Jul 31, 20221 min read

Molecular basis for ligand modulation of the cannabinoid CB 1 receptor

August 2022 "The cannabinoid CB1 receptor is the most abundant G protein coupled receptor (GPCR) in the central nervous system, which...

Dec 26, 20211 min read

G-protein-coupled receptors as therapeutic targets for glioblastoma

Glioblastoma multiforme (GBM) is the most common and aggressive primary brain tumour in adults. Treatments include surgical resection,...

Dec 1, 20211 min read

Obesity-induced changes in human islet G protein-coupled receptor expression: Implications for ...

Obesity-induced changes in human islet G protein-coupled receptor expression: Implications for metabolic regulation G protein-coupled...

Dec 1, 20211 min read

The development of modulators for lysophosphatidic acid receptors: A comprehensive review

Lysophosphatidic acids (LPAs) are bioactive phospholipids implicated in a wide range of cellular activities that regulate a diverse array...

Nov 1, 20211 min read

Genome-wide identification of 216 G protein-coupled receptor (GPCR) genes from the marine water ...

Genome-wide identification of 216 G protein-coupled receptor (GPCR) genes from the marine water flea Diaphanosoma celebensis G...