Identification of A2BAR as a potential target in colorectal cancer using novel fluorescent GPCR ligands "G-protein

Prokineticins (PKs) exert their biological functions through the activation of the G protein-coupled

AVPR2 is a kind of G protein coupled receptor (GPCR) and mainly couples with Gαs protein leading to cAMP

Significant advancements in the cellular biology of G protein-coupled receptors (GPCRs) about a novel

September 2022 "G protein‐coupled receptors (GPCRs) are valuable therapeutic targets for many diseases

September 2022 "G-protein-coupled receptors (GPCRs) are involved in a wide array of physiological and

Elucidation of a dynamic interplay between a beta-2 adrenergic receptor, its agonist, and stimulatory G Developing novel antifungals: lessons from G protein-coupled receptors.

November 2022 "Recently determined structures of class C G protein-coupled receptors (GPCRs) revealed

G-protein coupled receptors (GPCRs) play a paramount role in diverse brain functions.

β-arrestins (βarrs) play multifaceted roles in the function of G protein-coupled receptors (GPCRs). βarrs

radioligand binding assays with antibody-antigen interaction-based approaches for quantitative analysis of G

Pharmacological targeting of cGAS/STING-YAP signaling by both a small-molecule STING agonist, SR-717, and a G

G protein-coupled receptors (GPCRs) are critical myocardial signal transducers which regulate cardiac

Luciferase-based GloSensor™ cAMP assay: Temperature optimization and application to cell-based kinetic studies "G

X-ray crystallography, by cryo-EM has enabled insights into important drug target families such as G

critical component in multiple immune signaling processes and is dependent on activation by Ras and G

Currently, attention was mainly paid to biased signaling modulators targeting G protein-coupled receptors

Arrestins regulate a wide range of signaling events, most notably when bound to active G protein-coupled

G protein-coupled receptors (GPCRs) are among the most promising drug targets.

They recognize two types of G protein-coupled receptors (LPARs): LPA1-3 receptors and LPA4-6 receptors

GPR15 is a G protein-coupled receptor (GPCR) located on chromosome 3 and has similarity in its sequence

October 2022 "While the role of G-protein-coupled receptors (GPCR) in cancer is acknowledged, their underlying

The highest scoring protective hits included the complement C3a receptor (C3aR), a G-protein coupled

G protein-coupled receptor 3 (GPR3) belongs to the class A rhodopsin-type GPCR family and is highly expressed

forming a vicious cycle with IGF1/IGF1R signaling pathway "There is a potential correlation between G-protein-coupled

considered that TNBC is an estrogen-independent breast cancer, while a new estrogen receptor, namely G

amino acids, our current understanding on how endogenous PTHrP transduces signals through its cognate G-protein

Alterations in the expression and/or activity of brain G-protein-coupled receptors (GPCRs) such as dopamine