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249 items found for "homology modeling"
- The Impact of CB1 Receptor on Nuclear Receptors in Skeletal Muscle Cells
In conclusion, in skeletal muscle, CB1 receptors were recognized to be important moderators of NR4A1
- Constitutive, Basal, and β-Alanine-Mediated Activation of the Human Mas-Related G Protein-Coupled ..
coupled receptors (MRGPRs), a subfamily of GPCRs, are largely expressed by sensory neurons and known to modulate
- 📰 GPCR Weekly News, June 12 to 18, 2023
GPCR Activation and Signaling Single transmembrane GPCR modulating proteins: neither single nor simple
- An overview of the compartmentalized GPCR Signaling: Relevance and Implications
signaling has been extensively studied, highlighting their ability to scaffold various kinases and modulate stimulation of mitochondrial CB1 receptors by lipophilic agonists in these tissues was associated with the modulation
- 📰 GPCR Weekly News, August 7 to 13, 2023
GPCR Symposium on 'GPCRs as Therapeutic Modalities'. Want to share your project in a casual way?
- Enhancing GPCR Research Outreach | Dr GPCR University early-bird registration ends soon!
II Peptide Analogues: A Proposed Key Role of the N-Terminal Region for Novel Urotensin II Receptor Modulators
- 📰 GPCR Weekly News, May 22 to 28, 2023
Modulating GPCR and 14-3-3 protein interactions: prospects for CNS drug discovery.
- 📰 GPCR Weekly News, February 13 to 19, 2023
Structural and Molecular Insights into GPCR Function Quantitative analysis of sterol-modulated monomer-dimer
- 📰 GPCR Weekly News, August 14 to 20, 2023
GPCR Symposium on 'GPCRs as Therapeutic Modalities'.
- 📰 GPCR Weekly News, December 4 to 10, 2023
fundamental pharmacology in four weekly segments, delving into Agonists, Antagonists, and Allosteric Modulators
- 📰 GPCR Weekly News, April 3 to 9, 2023
SUCNR1 signaling in adipocytes controls energy metabolism by modulating circadian clock and leptin expression
- Therapeutic validation of an orphan G protein‐coupled receptor
IM (3,3′‐methylenebis‐1H‐indole) has been identified as a positive allosteric modulator of GPR84, a metabolite
- 📰 GPCR Weekly News, May 20 to 26, 2024
pathophysiological perspectives Structural and Molecular Insights into GPCR Function Bilayer lipids modulate
- 📰 GPCR Weekly News, September 25 to October 1, 2023
selectivity and is predominant for gene expression regulation by β2-adrenergic receptor Allosteric modulation probe dependence at Hydroxycarboxylic acid receptor HCAR2 Antipsychotic displays dual GPCR binding mode
- 📰 GPCR Weekly News, September 4 to 10, 2023
GPCR Symposium on ''GPCRs as Therapeutic Modalities' Share your project with a 1-minute abstract video
- 📰 GPCR Weekly News, May 8 to 14, 2023
An allosteric modulator of the adenosine A1 receptor potentiates the antilipolytic effect in rat adipose
- 📰 GPCR Weekly News, August 28 to September 3, 2023
GPCR Symposium on 'GPCRs as Therapeutic Modalities' Showcase your project with a 1-minute abstract video Binders, Drugs, and more The Leu/Val6.51 Side Chain of Cannabinoid Receptors Regulates the Binding Mode
- 📰 GPCR Weekly News, April 10 to 16, 2023
Reviews, GPCRs, and more Internal and external modulation factors of the orexin system (REVIEW).
- 📰 GPCR Weekly News, November 13 to 19, 2023
to a high salt challenge in the Dahl SS rat GPCRs in Neuroscience Neurokinin-2 receptor negatively modulates
- 📰 GPCR Weekly News, May 27 to June 2, 2024
effectively measure the strength of an allosteric effect as agonist's efficacy Single transmembrane GPCR modulating
- 📰 GPCR Weekly News, February 20 to 26, 2023
Allosteric modulation of conserved motifs and helices in 5HT2BR: Advances drug discovery and therapeutic
- 📰 GPCR Weekly News, April 15 to 21, 2024
GPCRs in Neuroscience Calcium-sensing receptor regulates Kv7 channels via Gi/o protein signalling and modulates
- 📰 GPCR Weekly News, February 12 to 18, 2024
agonism by Gαi/o-biased stapled peptide agonists of the relaxin-3 receptor GPCR kinases differentially modulate
- 📰 GPCR Weekly News, February 19 to 25, 2024
& Updates in GPCR Research A bioluminescent and homogeneous assay for monitoring GPCR-mediated cAMP modulation
- Ode to GPCRs
understanding of how various factors, such as lipid composition, osmotic stress, and allosteric ligands, modulate Interaction of G-Protein βγ Complex with Chromatin Modulates GPCR- Dependent Gene Regulation.