heterotrimeric G protein activity biosensors Marta Lopez-Balastegui , Antonella Di Pizio , Jiafei Mao , Jana Selent , et al. for their research on the Relevance of GPCR dynamics for receptor activation, signalling Principles of Pharmacology in Drug Discovery II -   Advanced Methods for the Optimization of Candidate Selection

work on Highly biased agonism for GPCR ligands via nanobody tethering Elk Kossatz, Michel Bouvier, Jana Selent, et al. for their study on G protein-specific mechanisms in the serotonin 5-HT2A receptor regulate pancreatic polypeptide from a structural, functional, and therapeutic perspective Structural basis for selectivity

October 2022 Structural perspectives on the mechanism of signal activation, ligand selectivity and allosteric opportunities to examine the dynamic fluxes in the 3D architecture of the receptors, as the basis of ligand selectivity Constituent structural motifs cooperatively transform ligand selectivity into specific functions, thus

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by targeting distinct subpockets of the orthosteric site Controlling the selectivity of aminergic GPCR small molecule agonists Two naturally occurring mutations of human GPR103 define distinct G protein selection for the Neuropeptides PACAP and VIP Coevolution underlies GPCR-G protein selectivity and functionality Site-selective labeling and electron paramagnetic resonance studies of human cannabinoid receptor CB2 modulated by different Dynorphin peptides First-Time Disclosure of CVN424, a Potent and Selective GPR6

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