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8 items found for "propionate"
- 📰 GPCR Weekly News, January 8 to 14, 2024
Receptor: Insights from Molecular Dynamics Simulations GPCRs in Cardiology, Endocrinology, and Taste Propionate
- Opioid Receptors and Protonation-Coupled Binding of Opioid Drugs
management could impact drug binding to the opioid receptor, because opioid drugs typically have a protonated amino group that contributes to receptor binding, and the functioning of GPCRs may involve protonation dynamics of opioid receptors from the perspective of the usefulness of computational studies to evaluate protonation-coupled
- AlphaFold2 versus experimental structures: evaluation on G protein-coupled receptors
However, a large portion of GPCR structures remain unsolved due to structural instability.
- Accelerating GPCR Drug Discovery With Conformation-Stabilizing VHHs
Despite this high number of GPCR targeted drugs, only a small portion (∼110) of the human GPCRome (consisting
- PAR-Induced Harnessing of EZH2 to β-Catenin: Implications for Colorectal Cancer
This methylation on a lysine residue at the N-terminal portion of β-catenin suppresses the ubiquitination
- 📰 GPCR Weekly News, November 6 to November 12, 2023
receptors GPCR Binders, Drugs, and more Discovery of (S)-3-(4-(benzyloxy)phenyl)-2-(2-phenoxyacetamido)propanoic
- 📰 GPCR Weekly News, January 30 to February 5, 2023
Valorization of leftover green tea residues through conversion to bioactive peptides using probiotics-aided
- Decoding β-Arrestins: from Structure to function
The "barcode hypothesis" proposes that β-arrestins decode distinct GPCR phosphorylation patterns, which Recent advancements in experimental and bioinformatics tools offer the potential to explore larger portions